| Irreversible inhibition of serine proteases by peptide derivatives of (. alpha.-aminoalkyl) phosphonate diphenyl esters J Oleksyszyn, JC Powers Biochemistry 30 (2), 485-493, 1991 | 254 | 1991 |
| Irreversible inhibition of serine proteases-design and in vivo activity of diaryl α-Aminophosphonate derivatives M Sienczyk, J Oleksyszyn Current medicinal chemistry 16 (13), 1673-1687, 2009 | 168 | 2009 |
| Dipeptide phosphonates as inhibitors of dipeptidyl peptidase IV B Boduszek, J Oleksyszyn, CM Kam, J Selzler, RE Smith, JC Powers Journal of medicinal chemistry 37 (23), 3969-3976, 1994 | 138 | 1994 |
| Diphenyl 1-aminoalkanephosphonates J Oleksyszyn, L Subotkowska, P Mastalerz | 137 | 1979 |
| Proline phosphonate derivatives JC Powers, B Boduszek, J Oleksyszyn US Patent 5,543,396, 1996 | 127 | 1996 |
| Novel amidine-containing peptidyl phosphonates as irreversible inhibitors for blood coagulation and related serine proteases J Oleksyszyn, B Boduszek, CM Kam, JC Powers Journal of medicinal chemistry 37 (2), 226-231, 1994 | 126 | 1994 |
| Comparision of the cytotoxic effects of birch bark extract, betulin and betulinic acid towards human gastric carcinoma and pancreatic carcinoma drug-sensitive and drug … M Drag, P Surowiak, M Drag-Zalesinska, M Dietel, H Lage, J Oleksyszyn Molecules 14 (4), 1639-1651, 2009 | 122 | 2009 |
| [30] Amino acid and peptide phosphonate derivatives as specific inhibitors of serine peptidases J Oleksyszyn, JC Powers Methods in enzymology 244, 423-441, 1994 | 111 | 1994 |
| Inhibition of Trypsin and Thrombin by Amino(4-amidinophenyl)methanephosphonate Diphenyl Ester Derivatives: X-ray Structures and Molecular Models, JA Bertrand, J Oleksyszyn, CM Kam, B Boduszek, S Presnell, RR Plaskon, ... Biochemistry 35 (10), 3147-3155, 1996 | 74 | 1996 |
| Irreversible inhibition of serine proteases by peptidyl derivatives of α-aminoalkylphosphonate diphenyl esters J Oleksyszyn, JC Powers Biochemical and biophysical research communications 161 (1), 143-149, 1989 | 65 | 1989 |
| Direct synthesis of 1-aminoalkanephosphonic and 1-aminoalkanephosphinic acids from phosphorus trichloride or dichlorophosphines J OLEKSYSZYN, T Roman, P MASTALERZ Synthesis 1978 (06), 479-480, 1978 | 63 | 1978 |
| Identification of a serine protease inhibitor which causes inclusion vacuole reduction and is lethal to Chlamydia trachomatis S Gloeckl, VA Ong, P Patel, JDA Tyndall, P Timms, KW Beagley, JA Allan, ... Molecular microbiology 89 (4), 676-689, 2013 | 60 | 2013 |
| Inhibition of trypsin and urokinase by Cbz-amino (4-guanidinophenyl) methanephosphonate aromatic ester derivatives: the influence of the ester group on their biological activity M Sieńczyk, J Oleksyszyn Bioorganic & medicinal chemistry letters 16 (11), 2886-2890, 2006 | 58 | 2006 |
| Human neutrophil elastase phosphonic inhibitors with improved potency of action £ Winiarski, J Oleksyszyn, M Sienczyk Journal of medicinal chemistry 55 (14), 6541-6553, 2012 | 57 | 2012 |
| Reaction of porcine pancreatic elastase with 7-substituted 3-alkoxy-4-chloroisocoumarins: design of potent inhibitors using the crystal structure of the complex formed with 4 … JC Powers, J Oleksyszyn, SL Narasimhan, CM Kam, R Radhakrishnan, ... Biochemistry 29 (12), 3108-3118, 1990 | 56 | 1990 |
| Expression of aminopeptidase N/CD13 in human ovarian cancers P Surowiak, M Dr±g, V Materna, S Suchocki, R Grzywa, M Spaczyński, ... International Journal of Gynecologic Cancer 16 (5), 2006 | 54 | 2006 |
| Mechanism-based isocoumarin inhibitors for human leukocyte elastase. Effect of the 7-amino substituent and 3-alkoxy group in 3-alkoxy-7-amino-4-chloroisocoumarins on inhibitory … JE Kerrigan, J Oleksyszyn, CM Kam, J Selzler, JC Powers Journal of medicinal chemistry 38 (3), 544-552, 1995 | 54 | 1995 |
| Plasminogen modulation of IL-1-stimulated degradation in bovine and human articular cartilage explants. The role of the endogenous inhibitors: PAI-1, α 2-antiplasmin, α 1-PI, α … J Oleksyszyn, AJ Augustine Inflammation Research 45, 464-472, 1996 | 46 | 1996 |
| New phosphonic analogs of aspartic and glutamic acid by aminoalkylation of trivalent phosphorus chlorides with ethyl acetyloacetate or ethyl levulinate and benzyl carbamate J Oleksyszyn, E Gruszecka, P Kafarski, P Mastalerz Monatshefte fuer Chemie Chemical Monthly 113 (1), 59-71, 1982 | 46 | 1982 |
| AN IMPROVED SYNTHESIS OF 1-AMINOPHOSPHONIC ACIDS. J Oleksyszyn, R Tyka | 44 | 1977 |
