Ewelina Węglarz-Tomczak
Ewelina Węglarz-Tomczak
University of Amsterdam, Swammerdam Institute for Life Sciences
Zweryfikowany adres z uva.nl - Strona główna
TytułCytowane przezRok
Azo dyes–biological activity and synthetic strategy
E Weglarz-Tomczak, L Gorecki
Chemik 66 (12), 1298-1307, 2012
512012
Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases
S Vassiliou, E Weglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, ...
Journal of medicinal chemistry 57 (19), 8140-8151, 2014
282014
A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases
E Węglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, A Joachimiak, ...
European journal of medicinal chemistry 117, 187-196, 2016
192016
Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues
E Węglarz-Tomczak, S Vassiliou, A Mucha
Bioorganic & medicinal chemistry letters 26 (16), 4122-4126, 2016
152016
An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and …
E Węglarz-Tomczak, M Poręba, A Byzia, Ł Berlicki, B Nocek, R Mulligan, ...
Biochimie 95 (2), 419-428, 2013
132013
An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and …
E Węglarz-Tomczak, M Poręba, ...
Biochimie 95 (2), 419-428, 2013
132013
Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and …
E Węglarz-Tomczak, M Burda-Grabowska, M Giurg, A Mucha
Bioorganic & medicinal chemistry letters 26 (21), 5254-5259, 2016
92016
Controlling the Helix Handedness of ααβ‐Peptide Foldamers through Sequence Shifting
M Szefczyk, E Węglarz‐Tomczak, P Fortuna, A Krzysztoń, ...
Angewandte Chemie International Edition 56 (8), 2087-2091, 2017
62017
Berlicki Ł, Pawełczak M, Nocek B, Mulligan R, Joachimiak A, Mucha A. Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and …
S Vassiliou, E Węglarz-Tomczak
J Med Chem 57, 8140-51, 2014
52014
Berlicki Ł, Nocek B, Mulligan, Joachimiak A, Drąg M, Mucha A. An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by …
E Węglarz-Tomczak, M Poręba, A Byzia
Biochimie 95 (2), 419-428, 2013
52013
Enantiomeric α, β-diaminoethylphosphonic acids as potent inhibitors of aminopeptidases—stereoselective synthesis and biological activity
E Węglarz-Tomczak, K Staszewska, M Talma, A Mucha
Tetrahedron Letters 57 (43), 4812-4814, 2016
32016
Estimating kinetic constants in the Michaelis–Menten model from one enzymatic assay using Approximate Bayesian Computation
JM Tomczak, E Węglarz‐Tomczak
FEBS letters 593 (19), 2742-2750, 2019
12019
Helix-loop-helix peptide foldamers and their use in the construction of hydrolase mimetics
M Drewniak, E Węglarz-Tomczak, K Ożga, E Rudzińska-Szostak, ...
Bioorganic chemistry 81, 356-361, 2018
12018
Barwniki azowe–aktywność biologiczna i strategie syntezy
E Węglarz-Tomczak, Ł Górecki
Chemik 66 (12), 2012
12012
Nature and Nurture integrated through an adjustable Flux Balance Analysis: The impact of cell-nutrition changes on the Warburg effect in hepatocellular carcinoma
E Węglarz-Tomczak, T Mondeel, DGE Piebes, HV Westerhoff
bioRxiv, 674150, 2019
2019
Neutral metalloaminopeptidases APN and MetAP2 as newly discovered anticancer molecular targets of actinomycin D and its simple analogs
E Węglarz-Tomczak, M Talma, M Giurg, HV Westerhoff, R Janowsk, ...
Oncotarget 9 (50), 29365-29378, 2018
2018
RATIONAL DESIGN, SYNTHESIS AND EVALUATION OF CATALYTICALLY ACTIVE PEPTIDE FOLDAMERS
L Berlicki, P Wojcik, M Szefczyk, M Drewniak, K Ozga, ...
JOURNAL OF PEPTIDE SCIENCE 22, S20-S20, 2016
2016
P1 AND P1'MODIFIED PHOSPHINIC DIPEPTIDE ANALOGUE INHIBITORS OF METALLOAMINOPEPTIDASES
M Talma, E Weglarz-Tomczak, K Staszewska, A Mucha
JOURNAL OF PEPTIDE SCIENCE 22, S184-S184, 2016
2016
Inhibition of Neisseria meningitidis Alanine Aminopeptidase with Phosphinic Dipeptide Analogs
A Mucha, S Vassiliou, E Weglarz-Tomczak, L Berlicki, M Paweiczak, ...
BIOPOLYMERS 100 (3), 306-306, 2013
2013
NOVEL PHOSPHORUS-CONTAINING AMINO ACID AND DIPEPTIDE MIMETICS AS HIGHLY POTENT INHIBITORS OF NEISSERIA MENINGITIDIS ALANYL AMINOPEPTIDASE
E Węglarz-Tomczak, S Vassiliou, Ł Berlicki, M Pawełczak, B Nocek, ...
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