The C loop at the orthosteric binding site is critically involved in GABAA receptor gating K Terejko, PT Kaczor, MA Michałowski, A Dąbrowska, JW Mozrzymas Neuropharmacology 166, 107903, 2020 | 20 | 2020 |
Distinct Modulation of Spontaneous and GABA-Evoked Gating by Flurazepam Shapes Cross-Talk Between Agonist-Free and Liganded GABAA Receptor Activity M Jatczak-Śliwa, K Terejko, M Brodzki, MA Michałowski, MM Czyzewska, ... Frontiers in Cellular Neuroscience 12, 237, 2018 | 15 | 2018 |
Mutations of α1F45 residue of GABAA receptor loop G reveal its involvement in agonist binding and channel opening/closing transitions M Brodzki, MA Michałowski, M Gos, JW Mozrzymas Biochemical Pharmacology 177, 113917, 2020 | 11 | 2020 |
Binding site opening by loop C shift and chloride ion-pore interaction in the GABA A receptor model MA Michałowski, S Kraszewski, JW Mozrzymas Physical Chemistry Chemical Physics 19 (21), 13664-13678, 2017 | 11 | 2017 |
Interaction between GABAA receptor α1 and β2 subunits at the N-terminal peripheral regions is crucial for receptor binding and gating K Terejko, MA Michałowski, A Dominik, A Andrzejczak, JW Mozrzymas Biochemical Pharmacology 183, 114338, 2021 | 9 | 2021 |
α1 Proline 277 Residues Regulate GABAAR Gating through M2-M3 Loop Interaction in the Interface Region PT Kaczor, MA Michałowski, JW Mozrzymas ACS Chemical Neuroscience 13 (21), 3044-3056, 2022 | 7 | 2022 |
Mutations at the M2 and M3 Transmembrane Helices of the GABAARs α1 and β2 Subunits Affect Primarily Late Gating Transitions Including Opening/Closing and … K Terejko, MA Michałowski, I Iżykowska, A Dominik, A Brzóstowicz, ... ACS Chemical Neuroscience 12 (13), 2421-2436, 2021 | 6 | 2021 |
Mutation of valine 53 at the interface between extracellular and transmembrane domains of the β2 principal subunit affects the GABAA receptor gating K Kłopotowski, MA Michałowski, M Gos, D Mosiądz, MM Czyżewska, ... European Journal of Pharmacology 947, 175664, 2023 | 1 | 2023 |
The β2 subunit E155 residue as a proton sensor at the binding site on GABA type A receptors MA Michałowski, MM Czyżewska, I Iżykowska, JW Mozrzymas European Journal of Pharmacology 906, 174293, 2021 | 1 | 2021 |
Neuropharmaco ogy K Terejko, PT Kaczor, MA Michałowski, A Dąbrowska, JW Mozrzymas Neuropharmacology 166, 107903, 2020 | | 2020 |