Obserwuj
Paweł Zajdel
Paweł Zajdel
Jagiellonian University Medical College
Zweryfikowany adres z uj.edu.pl
Tytuł
Cytowane przez
Cytowane przez
Rok
Antidepressant and antipsychotic activity of new quinoline-and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT1A/5-HT2A/5-HT7 and dopamine D2/D3 receptors
P Zajdel, K Marciniec, A Maślankiewicz, K Grychowska, G Satała, ...
European Journal of Medicinal Chemistry 60, 42-50, 2013
932013
Quinoline-and isoquinoline-sulfonamide analogs of aripiprazole: novel antipsychotic agents?
P Zajdel, A Partyka, K Marciniec, AJ Bojarski, M Pawlowski, ...
Future medicinal chemistry 6 (1), 57-75, 2014
892014
Physical interaction between neurofibromin and serotonin 5-HT6 receptor promotes receptor constitutive activity
W Deraredj Nadim, S Chaumont-Dubel, F Madouri, L Cobret, ...
Proceedings of the National Academy of Sciences 113 (43), 12310-12315, 2016
872016
Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with …
K Grychowska, G Satała, T Kos, A Partyka, E Colacino, ...
ACS Chemical Neuroscience 7 (7), 972-983, 2016
782016
Imidazopyridine-based selective and multifunctional ligands of biological targets associated with psychiatric and neurodegenerative diseases
D Vanda, P Zajdel, M Soural
European Journal of Medicinal Chemistry 181, 111569, 2019
682019
Quinoline-and isoquinoline-sulfonamide derivatives of LCAP as potent CNS multi-receptor—5-HT1A/5-HT2A/5-HT7 and D2/D3/D4—agents: The synthesis and pharmacological evaluation
P Zajdel, K Marciniec, A Maślankiewicz, G Satała, B Duszyńska, ...
Bioorganic & medicinal chemistry 20 (4), 1545-1556, 2012
652012
Separation and characterization of ciprofloxacin, difloxacin, lomefloxacin, norfloxacin, and ofloxacin oxidation products under potassium permanganate treatment in acidic …
U Hubicka, P Żmudzki, B Żuromska-Witek, P Zajdel, M Pawłowski, J Krzek
Talanta 109, 91-100, 2013
542013
Novel multi-target azinesulfonamides of cyclic amine derivatives as potential antipsychotics with pro-social and pro-cognitive effects
P Zajdel, T Kos, K Marciniec, G Satała, V Canale, K Kamiński, M Hołuj, ...
European Journal of Medicinal Chemistry 145, 790-804, 2018
472018
N1-Azinylsulfonyl-1H-indoles: 5-HT6 Receptor Antagonists with Procognitive and Antidepressant-Like Properties
P Zajdel, K Marciniec, G Satała, V Canale, T Kos, A Partyka, ...
ACS Medicinal Chemistry Letters 7 (6), 618-622, 2016
472016
The multiobjective based design, synthesis and evaluation of the arylsulfonamide/amide derivatives of aryloxyethyl-and arylthioethyl-piperidines and pyrrolidines as a novel …
P Zajdel, R Kurczab, K Grychowska, G Satała, M Pawłowski, AJ Bojarski
European journal of medicinal chemistry 56, 348-360, 2012
472012
Arene-and quinoline-sulfonamides as novel 5-HT7 receptor ligands
P Zajdel, K Marciniec, A Maślankiewicz, MH Paluchowska, G Satała, ...
Bioorganic & medicinal chemistry 19 (22), 6750-6759, 2011
442011
Novel non-sulfonamide 5-HT6 receptor partial inverse agonist in a group of imidazo [4, 5-b] pyridines with cognition enhancing properties
D Vanda, M Soural, V Canale, S Chaumont-Dubel, G Satała, T Kos, ...
European Journal of Medicinal Chemistry 144, 716-729, 2018
432018
Novel class of arylpiperazines containing N-acylated amino acids: Their synthesis, 5-HT1A, 5-HT2A receptor affinity, and in vivo pharmacological evaluation
P Zajdel, G Subra, AJ Bojarski, B Duszyńska, E Tatarczyńska, A Nikiforuk, ...
Bioorganic & medicinal chemistry 15 (8), 2907-2919, 2007
402007
A New Class of Arylpiperazine Derivatives:  the Library Synthesis on SynPhase Lanterns and Biological Evaluation on Serotonin 5-HT1A and 5-HT2A Receptors
P Zajdel, G Subra, AJ Bojarski, B Duszyńska, M Pawłowski, J Martinez
Journal of Combinatorial Chemistry 6 (5), 761-767, 2004
402004
From haloquinolines and halopyridines to quinoline-and pyridinesulfonyl chlorides and sulfonamides
A Maslankiewicz, K Marciniec, M Pawlowski, P Zajdel
Heterocycles 71 (9), 1975-1990, 2007
392007
New Arylpiperazine 5-HT1A Receptor Ligands Containing the Pyrimido[2,1-f]purine Fragment:  Synthesis, in Vitro, and in Vivo Pharmacological Evaluation
S Jurczyk, M Kołaczkowski, E Maryniak, P Zajdel, M Pawłowski, ...
Journal of medicinal chemistry 47 (10), 2659-2666, 2004
392004
Towards new 5-HT7 antagonists among arylsulfonamide derivatives of (aryloxy) ethyl-alkyl amines: multiobjective based design, synthesis, and antidepressant and anxiolytic …
V Canale, R Kurczab, A Partyka, G Satała, T Lenda, ...
European journal of medicinal chemistry 108, 334-346, 2016
382016
Ergotamine and nicergoline—facts and myths
P Zajdel, M Bednarski, J Sapa, G Nowak
Pharmacological Reports 67, 360-363, 2015
342015
Amino Acid Hot Spots of Halogen Bonding: A Combined Theoretical and Experimental Case Study of the 5-HT7 Receptor
R Kurczab, V Canale, G Satała, P Zajdel, AJ Bojarski
Journal of Medicinal Chemistry 61 (19), 8717-8733, 2018
332018
Virtual screening-driven discovery of dual 5-HT6/5-HT2A receptor ligands with pro-cognitive properties
J Staroń, R Kurczab, D Warszycki, G Satała, M Krawczyk, R Bugno, ...
European Journal of Medicinal Chemistry 185, 111857, 2020
322020
Nie można teraz wykonać tej operacji. Spróbuj ponownie później.
Prace 1–20