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Vimal Varghese
Vimal Varghese
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Cited by
Year
Structural and functional insight into human O-GlcNAcase
C Roth, S Chan, WA Offen, GR Hemsworth, LI Willems, DT King, ...
Nature chemical biology 13 (6), 610-612, 2017
1082017
NHC catalyzed transformation of aromatic aldehydes to acids by carbon dioxide: an unexpected reaction
V Nair, V Varghese, RR Paul, A Jose, CR Sinu, RS Menon
Organic Letters 12 (11), 2653-2655, 2010
1082010
Nucleophilic heterocyclic carbene catalyzed annulation of enals to chalcones in methanol: a stereoselective synthesis of highly functionalized cyclopentanes
V Nair, BP Babu, S Vellalath, V Varghese, AE Raveendran, E Suresh
Organic Letters 11 (12), 2507-2510, 2009
972009
Novel nucleophilic heterocyclic carbene mediated stereoselective conjugate addition of enals to nitrostyrenes via homoenolate
V Nair, CR Sinu, BP Babu, V Varghese, A Jose, E Suresh
Organic Letters 11 (24), 5570-5573, 2009
882009
Short Chemoenzymatic Total Synthesis of ent‐Hydromorphone: An Oxidative Dearomatization/Intramolecular [4+2] Cycloaddition/Amination Sequence
V Varghese, T Hudlicky
Angewandte Chemie International Edition 53 (17), 4355-4358, 2014
692014
A convenient approach to stereoisomeric iminocyclitols: generation of potent brain‐permeable OGA inhibitors
M Bergeron‐Brlek, J Goodwin‐Tindall, N Cekic, C Roth, WF Zandberg, ...
Angewandte Chemie International Edition 54 (51), 15429-15433, 2015
472015
A novel pseudo four component reaction involving homoenolate for the synthesis of γ-aminobutyric acid (GABA) derivatives
V Nair, V Varghese, BP Babu, CR Sinu, E Suresh
Organic & Biomolecular Chemistry 8 (4), 761-764, 2010
452010
Total synthesis of dihydrocodeine and hydrocodone via a double Claisen rearrangement and C-10/C-11 closure strategy
V Varghese, T Hudlicky
Synlett 24 (03), 369-374, 2013
312013
A novel multicomponent reaction involving isoquinoline, allenoate and cyanoacrylates
V Nair, BP Babu, V Varghese, CR Sinu, RR Paul, ER Anabha, E Suresh
Tetrahedron Letters 50 (26), 3716-3718, 2009
302009
NHC-catalysed annulation of enals to tethered dienones: efficient synthesis of bicyclic dienes
V Nair, S Vellalath, BP Babu, V Varghese, RR Paul, E Suresh
Organic & Biomolecular Chemistry 8 (21), 4861-4866, 2010
272010
Processes for preparing ACC inhibitors and solid forms thereof
M Geier, N Ikemoto, S Liew, ME Scott, V Varghese
US Patent 10,519,165, 2019
102019
Solid forms of a thienopyrimidinedione ACC inhibitor and methods for production thereof
S Calimsiz, M Geier, GC Harriman, JP Lawson, K Sabourin, ME Scott, ...
US Patent 10,487,090, 2019
102019
A short history of the discovery and development of naltrexone and other morphine derivatives
V Varghese, T Hudlicky
Natural Products in Medicinal Chemistry 60, 225-250, 2014
92014
Nitrone cycloaddition to quinones: A novel strategy for the synthesis of benzisoxazolidenes
RR Paul, V Varghese, PB Beneesh, CR Sinu, E Suresh, ER Anabha
Journal of Heterocyclic Chemistry 47 (2), 396-399, 2010
32010
Solid forms of a thienopyrimidinedione acc inhibitor and methods for production thereof
K Alexander, JC Amedio, S Calimsiz, M Geier, GC Harriman, S Hu, ...
US Patent App. 17/393,030, 2022
2*2022
Cover Picture: Short Chemoenzymatic Total Synthesis of ent‐Hydromorphone: An Oxidative Dearomatization/Intramolecular [4+2] Cycloaddition/Amination …
V Varghese, T Hudlicky
Angewandte Chemie International Edition 53 (17), 4251-4251, 2014
22014
Processes for preparing acc inhibitors and solid forms thereof
M Geier, L Humphreys, N Ikemoto, S Liew, H Morrison, ME Scott, ...
US Patent App. 16/924,924, 2021
2021
Process for preparing morphine compounds
V Varghese, T Hudlicky
US Patent 9,126,965, 2015
2015
Chemoenzymatic Total Synthesis of Morphine alkaloids: Synthesis of Dihydrocodeine and Hydrocodone via a Double Claisen Strategy and ent-Hydromorphone via an Oxidative …
V Varghese
Brock University, 2015
2015
Titelbild: Short Chemoenzymatic Total Synthesis of ent‐Hydromorphone: An Oxidative Dearomatization/Intramolecular [4+ 2] Cycloaddition/Amination Sequence (Angew. Chem. 17/2014)
V Varghese, T Hudlicky
Angewandte Chemie 126 (17), 4337-4337, 2014
2014
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